Nitric Oxide Releasing Rosiglitazone Derivatives:Design,Synthesis and Biological Evaluation

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户:ZHUZHU1987251
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  Rosiglitazone is clinically used to treat insulin resistance.However,its long-term administration will increase the incidence of cardiovascular side effects.[1] Given the beneficial effects of nitric oxide(NO)on endothelial function as an anti-hypertensive agent[2],we are motivated to synthesize hybrid compounds of rosiglitazone bearing nitrate-or diazeniumdiolate-based NO donating moieties.
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