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5. Synthesis of Benzimidazole-based Fluconazole Analogues and Relational Antimicrobial Evaluation

Synthesis of Benzimidazole-based Fluconazole Analogues and Relational Antimicrobial Evaluation

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户：forsanwang

【摘 要】

：

Fluconazole is a well known first-line antifungal drug recommended by World Health Organization and is prevalently used to treat fungal infections by Candida albicans and Cryptococcus neoformans with

【作 者】

：

Shi-Chao HE Jeyakkumar PONMANI Hui-Zhen ZHANG Cheng-He ZHOU 

【机 构】

：

Laboratory of Bioorganic & Medicinal Chemistry,School of Chemistry and Chemical Engineering,Southwes

【出 处】

：

2015年全国药物化学学术会议暨第五届中英药物化学学术会议

【发表日期】

：

2015年3期

【关键词】

：

Benzimidazole Fluconazole Antibacterial Antifungal 

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论文部分内容阅读

　　Fluconazole is a well known first-line antifungal drug recommended by World Health Organization and is prevalently used to treat fungal infections by Candida albicans and Cryptococcus neoformans with an exceptional therapeutic record including good activity and favourable pharmacokinetic characteristics.

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