Atom-Economic Synthesis of Fully Substituted 2-Aminopyrroles via Gold-Catalyzed Formal [3+2] Cycload

来源 :中国化学会第九届全国有机化学学术会议 | 被引量 : 0次 | 上传用户:zhq198709
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As part of our continuous efforts to study on the ynamide chemistry,we describe herein a novel gold-catalyzed formal [3+2] cycloaddition between ynamides and fully substituted isoxazoles,leading to the concise and efficient synthesis of various fully substituted 2-aminopyrroles.
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