大黄素对重症胰腺炎肾损伤模型大鼠血清缺氧诱导因子-1α及糖原合酶激酶-3β水平的影响

来源 :中国临床药理学杂志 | 被引量 : 0次 | 上传用户:yezhenhao
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
目的研究大黄素对重症胰腺炎肾损伤大鼠血清缺氧诱导因子-1α(HIF-1α)和糖原合酶激酶-3β(GSK-3β)水平影响。方法将60只大鼠随机分为空白组、假手术组、模型组、对照组和实验组,每组12只。模型组和试验组注入牛磺胆酸钠0.1 mL/100 g建立重症胰腺炎肾损伤大鼠模型;假手术组和对照组打开腹腔后仅轻轻翻动十二指肠以及胰腺;空白组大鼠未作任何处理。空白组、假手术组、模型组均予以腹腔注射5μL·g-10.9%Na Cl q6 h;对照组和实验组均按25μg·g-1剂量予以腹腔注射5 g·L~(-1)大黄素q6 h。术后3,6,12h,比较各组大鼠的血清肌酸酐(SCr)、尿素氮(BUN)、HIF-1α和GSK-3β水平。结果空白组、假手术组、对照组和实验组的胰腺组织病理学评分分别为(1.30±0.14),(1.39±0.14),(1.40±0.15)和(2.73±0.30)分,与模型组的胰腺组织病理学评分(9.84±1.05)分相比,差异均有统计学意义(均P<0.05),且实验组的胰腺组织病理学评分与空白组、假手术组、对照组比较,差异均有统计学意义(均P<0.05)。术后3 h,空白组、假手术组、对照组、模型组和实验组的SCr分别为(60.46±6.78),(61.52±6.78),(60.38±6.74),(120.57±13.43)和(95.35±9.85)μmol·L~(-1),BUN分别为(7.47±0.79),(8.02±0.92),(7.93±0.83),(12.49±1.53)和(8.56±0.89)mmol·L~(-1),HIF-1α分别为(225.46±23.57),(210.57±23.58),(229.67±6.74),(160.46±17.47)和(144.57±14.85)μg·L~(-1),GSK-3β分别为(6.59±0.69),(6.57±0.69),(6.74±0.68),(19.95±2.13)和(10.56±1.39)μg·L~(-1)。术后6 h,空白组、假手术组、对照组、模型组和实验组的SCr分别为(60.57±6.79),(60.55±6.76),(59.50±6.76),(143.57±15.47)和(110.57±12.55)μmol·L~(-1),BUN分别为(7.65±0.84),(8.11±0.93),(8.29±0.92),(15.46±1.64)和(12.35±1.37)mmol·L~(-1),HIF-1α分别为(226.46±24.04),(222.46±23.57),(230.57±24.05),(155.36±15.74)和(127.57±12.84)μg·L~(-1),GSK-3β分别为(6.25±0.67),(6.71±0.69),(6.82±0.71),(25.34±2.64)和(11.56±1.27)μg·L~(-1)。术后12 h,空白组、假手术组、对照组、模型组和实验组的SCr分别为(60.61±6.79),(61.68±6.79),(61.54±6.78),(166.45±17.05)和(131.45±13.46)μmol·L~(-1),BUN分别为(8.03±0.85),(7.98±0.82),(8.79±0.93),(18.66±19.46)和(15.35±1.63)mmol·L~(-1),HIF-1α分别为(219.57±23.63),(226.35±24.04),(220.25±24.04),(148.46±18.94)和(117.46±12.04)μg·L~(-1),GSK-3β分别为(6.77±0.69),(6.70±0.70),(6.86±0.70),(35.02±3.76)和(20.35±2.13)μg·L~(-1)。空白组、假手术组、对照组术后3,6,12 h的SCr、BUN、HIF-1α、GSK-3β与模型组比较,差异均有统计学意义(均P<0.05),且实验组与模型组术后3,6,12 h的SCr、BUN、HIF-1α、GSK-3β比较,差异均有统计学意义(均P<0.05)。结论大黄素可能通过上调血清HIF-1α和GSK-3β水平,提高肾细胞耐缺氧的能力,从而发挥对重症急性胰腺炎肾损伤的保护作用。 Objective To investigate the effects of emodin on serum levels of hypoxia inducible factor-1α (HIF-1α) and glycogen synthase kinase-3β (GSK-3β) in rats with severe pancreatitis and renal injury. Methods Sixty rats were randomly divided into blank group, sham operation group, model group, control group and experimental group, with 12 rats in each group. Model group and experimental group were infused with sodium taurocholate 0.1 mL / 100 g to establish a rat model of severe acute pancreatitis and renal injury. The rats in sham-operated group and control group were gently inflected to open duodenum and pancreas, Without any treatment. The rats in the blank group, sham operation group and model group were intraperitoneally injected with 5 μL · g-10.9% NaCl q for 6 h. The control group and experimental group were injected intraperitoneally with 5 g · L -1 rhubarb Prime q6 h. Serum creatinine (SCr), blood urea nitrogen (BUN), HIF-1α and GSK-3β levels were compared between the three groups at 3, 6 and 12 h after operation. Results The histopathological scores of pancreatic tissue in the blank group, the sham operation group, the control group and the experimental group were (1.30 ± 0.14), (1.39 ± 0.14), (1.40 ± 0.15) and (2.73 ± 0.30) There were significant differences between the two groups (all P <0.05), and the difference of pancreatic histopathological score between the experimental group and the blank group, the sham operation group and the control group were statistically significant There was statistical significance (all P <0.05). The SCr of the blank group, the sham operation group, the control group, the model group and the experimental group were (60.46 ± 6.78), (61.52 ± 6.78), (60.38 ± 6.74), (120.57 ± 13.43) and (95.35 ± 9.85) μmol·L -1, BUN were (7.47 ± 0.79), (8.02 ± 0.92), (7.93 ± 0.83), (12.49 ± 1.53) and (8.56 ± 0.89) mmol·L ~ 1 and HIF-1α were (225.46 ± 23.57), (210.57 ± 23.58), (229.67 ± 6.74), (160.46 ± 17.47) and (144.57 ± 14.85) μg · L -1, respectively (6.59 ± 0.69), (6.57 ± 0.69), (6.74 ± 0.68), (19.95 ± 2.13) and (10.56 ± 1.39) μg · L -1, respectively. The SCr of the blank group, the sham operation group, the control group, the model group and the experimental group were (60.57 ± 6.79), (60.55 ± 6.76), (59.50 ± 6.76), (143.57 ± 15.47) and (110.57 ± 12.55) μmol·L -1, BUN were (7.65 ± 0.84), (8.11 ± 0.93), (8.29 ± 0.92), (15.46 ± 1.64) and (12.35 ± 1.37) mmol·L -1 1 and HIF-1α were (226.46 ± 24.04), (222.46 ± 23.57), (230.57 ± 24.05), (155.36 ± 15.74) and (127.57 ± 12.84) μg · L -1, respectively (6.25 ± 0.67), (6.71 ± 0.69), (6.82 ± 0.71), (25.34 ± 2.64) and (11.56 ± 1.27) μg · L -1, respectively. The SCr of the blank group, the sham operation group, the control group, the model group and the experimental group were (60.61 ± 6.79), (61.68 ± 6.79), (61.54 ± 6.78), (166.45 ± 17.05) and (131.45 ± 13.46μmol·L -1 and BUN were respectively (8.03 ± 0.85), (7.98 ± 0.82), (8.79 ± 0.93), (18.66 ± 19.46) and (15.35 ± 1.63) mmol·L ~ (-1) 1 and HIF-1α were (219.57 ± 23.63), (226.35 ± 24.04), (220.25 ± 24.04), (148.46 ± 18.94) and (117.46 ± 12.04) μg · L -1, respectively (6.77 ± 0.69), (6.70 ± 0.70), (6.86 ± 0.70), (35.02 ± 3.76) and (20.35 ± 2.13) μg · L -1, respectively. The levels of SCr, BUN, HIF-1α and GSK-3β in the blank group, the sham operation group and the control group at 3, 6 and 12 h postoperatively were significantly different from those in the model group (all P <0.05) Compared with model group, SCr, BUN, HIF-1α and GSK-3β at 3, 6 and 12 h after operation were significantly different (all P <0.05). Conclusion Emodin may play a protective role in renal injury induced by severe acute pancreatitis by up-regulating the serum levels of HIF-1α and GSK-3β and increasing the hypoxic tolerance of renal cells.
其他文献
听力是英语学习者必须要掌握的四项基本技能(听、说、读、写)之一,也是英语学习者认为比较难的技能之一,而词汇是英语学习的前提条件。本研究以Nation(1990)的词汇知识理论框
全球经济一体化和电子商务的飞速发展,更加凸显了英语作为世界性语言的地位,商务英语发展成为专门用途英语最重要的一个分支。随着我国高等职业技术教育的快速发展,全国各地
针对分布式的松散耦合的多系统构成的数字图书馆服务体系,提出基于应用层的数字图书馆网络服务监测方案,实现可访问即可监测的服务管理目标,并给出服务性能预警和可用性的计算方
介绍基于模式自动机的全文检索系统的工作原理、体系结构,并给出基于模式自动机的全文索引数据库的核心数据结构和相关的生成算法、检索算法和模式自学习算法。
在过去的几十年里,二语交易意愿吸引了来自二语习得领域专家学者们的诸多目光。研究者们认为,外语学习应更注重语言实际应用而非应试能力,因此学生是否能够愿意与他人进行目
当今世界,全球交流日趋频繁,各国高层领导人频频出席国际场合,发表演说。口译在整个过程中则发挥着举足轻重的作用,为具备不同文化背景的人群扫除语言障碍,以达到相互理解的
抗抑郁药已在临床上应用了几十年,然而直到现在抗抑郁药的作用机制还不清楚。越来越多的研究表明抗抑郁治疗能够增加神经营养因子的表达水平和调节海马内神经发生,并且抗抑郁
对于初中生而言,错题整理是“甜蜜的负担”。教师对错题本的认可是学生心中“甜蜜的期待”。但是在整理的过程中,没有规范的指引和激励措施,学生会感到压力很大。所以,本文以
本报告是在目的论指导下,基于《英语学术论文写作》(第四章)英译汉的翻译实践完成的。以目的论的三原则为指导,并根据原文本的相关特点,译者采取不同的翻译策略,实现目的语翻
张爱玲(1920-1995)是20世纪中国文学史上著名的女性作家,也是为数不多的可以纯熟自由地运用双语写作与翻译,并取得一定声誉的作家之一。她对自己作品的翻译从20世纪50年代开