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４－（２－氨乙基）吗啉（１）是重要的医药中间体及有机合成原料。主要通过下列几种方法合成：ａ）以吗啉为原料。用２－氯乙胺［１］、２－溴乙胺［２］或氮丙啶［３］和吗啉进行缩合；用３－吗啉基丙酰胺［４］与次氯酸钠反应；或由２－吗啉基乙酰胺［５］、２－吗啉基...
4- (2-aminoethyl) morpholine (1) is an important pharmaceutical intermediates and organic synthesis of raw materials. Mainly through the following methods of synthesis: a) Morpholine as raw material. Condensation with 2-chloroethylamine [1], 2-bromoethylamine [2] or aziridine [3] and morpholine; reaction with sodium hypochlorite with 3- morpholinopropionamide [4] Morpholinyl acetamide [5], 2-morpholino ...