imidazo[1相关论文
Micellar Catalysis:Visible-Light Mediated Imidazo[1,2-a]pyridine C—H Amination with N-Aminopyridiniu
A light-promoted metal-free protocol for the amination of imidazo[1,2-a]pyridines with N-aminopyridinium salt by the ass......
The widespread applications of aggregation-induced emission luminogens (AIEgens) inspire the creation of AIEgens with no......
Design,synthesis and biological evaluation of novel imidazo[1,2-a]pyridine derivatives as potent ant
Antimitotic drugs play an important role in anti-tumor treatment,and various new scaffords of Tubulin inhibitors have be......
Design,Synthesis,and Biological Evaluation of Novel Imidazo[1,2-a]pyridine Derivatives as Potent c-M
A series of imidazo[1,2-a]pyridine derivatives against c-Met was designed by means of bioisosteric replacement.1 In our ......
The mammalian target of rapamycin(mTOR)is a critical component part of the PI3K-Akt signaling pathway that plays a key r......
Synthesis and Catalytic Application in Transfer Hydrogenation of 2,6-Bis(imidazo[1,2-a]pyridin-2-yl)
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Metal-free Oxidative Coupling of Aminopyridines with Nitroolefins to Imidazo[1,2-a]pyridine in the P
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Luminescent transition metal complexes have attracted great attention due to their various applications,such as in organ......
Imidazopyridine are classes of fused heterocycles that are of considerable interest because of the diverse range of thei......
Catalyst-Free Friedel-Crafts Hydroxyalkylation of Imidazo[1,2-α]pyridines with Ethyl Trifluoropyruva
Remarkable developments have been made on the synthesis of imidazo[1,2-α]pyridine derivatives,[1] making a wide range o......
Imidazopyridine compounds are important nitrogen-containing heterocycles existing widely in natural products,pharmaceuti......
The 1,2,3-triazole scaffold plays an important role in medicinal arena as numerous molecules bearing this framework are ......
发展了一个无光敏剂参与的可见光促进的咪唑并[1,2-a]吡啶衍生物的三氟甲基化新反应.该反应利用本课题组此前发展的基于硫叶立德骨......
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咪唑并吡啶[1,5-a]类化合物是一类具有环合氮类的杂环化合物,在自然界中并不广存在.但是近些年来的研究发现,这类杂环包括它的衍生......
本文通过对荣华二采区10...
Abnormal Nucleophilic Reaction of Ethyl Crotonate: An Easy Way to Form Novel Imidazo[1,5-a] pyridine
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Synthesis and Evaluation of 8-[131I]Iodo-substituted Imidazopyridine Derivative as Single Photon Emi
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
以异噁唑啉基环取代呋喃核糖环(ribose ring)为基本单元,成功地合成了一系列咪唑[1,2-a]吡啶衍生物的C-核苷化合物3和4(其中碱基和......
Abnormal Nucleophilic Reaction of Ethyl Crotonate: An Easy Way to Form Novel Imidazo[1,5-a] pyridine
An abnormal intramolecular nucleophilic reaction of α-carbon of α,β-unsaturated ester was discovered and the reaction......
Synthesis and Evaluation of 8-[131I]Iodo-substituted Imidazopyridine Derivative as Single Photon Emi
A novel N-methyl, N-phenyl-[6-chloro-2-(4-chlorophenyl)-8-iodoimidazo[1, 2-a]-pyridine-3-yl]acetamide (compound Ⅴ) was ......
本文报道CLINDE改进的合成方法及其同位素^131I-标记。标记前体由5-氯-2-氨基吡啶与溴代酮酰胺缩合制得。标记产物经三烷基锡化、......
以联苯胺为原料,通过三组份串联反应一步合成咪唑[1,5-a]吡啶型离子(L),其结构经1H NMR,13C NMR,IR和X-射线单晶衍射表征。利用荧光......
醌构咪唑并[1,2-a]吡啶类化合物是具有广泛生物活性的一类化合物。研究了1,4-萘醌与2-氨基吡啶经钯催化的C—H键乙酰化过程的环合......
以6-氨基-3-吡啶甲酸为起始原料,经过酯化反应、环合反应、还原反应得到7-羟甲基咪唑并[1,2-a]吡啶,总收率为42%.......
Reaction of Nitrilimines with 2-Aminopicoline, 3-Amino-1,2,4-Triazole, 5-Aminotetrazole and 2-Aminop
The reaction of picoline derivatives 3-6 with hydrazonoylhalide 1a produced imidazo[1,2-a]pyridines 7-10, while the reac......
分别在常规加热和微波辐射条件下,由双(2-吡啶甲酰)、二(2-吡啶)甲酮与脂肪醛及醋酸铵在醋酸溶剂中反应成功地制备了3-烷基取代的咪唑并......
一系列 imidazo [1,2-a ] 嘧啶衍生物在位置与二芳基邻近地代替了 2 和 3 被设计并且综合了以便改进他们的反煽动性的活动。生物测......
Synthesis and Evaluation of 8-[^131I]Iodo-substituted Imidazopyridine Derivative as Single Photon Em
<正>A novel N-methyl, N-phenyl-[6-chloro-2-(4-chlorophenyl)-8-iodoimidazo[1, 2-α]-pyridine-3-yl]acetamide (compoundⅤ) ......
目的:基于氧化碳氢键官能团化策略,重新构建咪唑并[1,5-a]吡啶的合成方法。方法:以2-苄基吡啶和苄胺为反应原料,采用单因素试验法,考......
CuⅡ and CuⅠ Complexes of 1,1'-(Pyridin-2-ylmethylene)-bis[3-(pyridin-2-yl)imidazo[1,5-a]pyridine]:in
Reaction of 3-(pyridin-2-yl)-imidazo[1,5-a]pyridine(HPIP), Cu Cl2·2H2O and picolinaldehyde in the mixture of CH3 CO......
A one-pot three component condensation synthesis of imidazo[1,5-a]pyridines using of various aromatic aldehydes and dipy......