【摘 要】
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Quinoxalines are an important class of nitrogen-containing heterocyclesthat possess a broad spectrum of physiological and biological activities.1 Although a number of methods are available for the syn
【机 构】
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State Key Laboratory of Elemento-Organic Chemistry, Institute of Elemento-Organic Chemsitry, Nankai
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Quinoxalines are an important class of nitrogen-containing heterocyclesthat possess a broad spectrum of physiological and biological activities.1 Although a number of methods are available for the synthesis of racemic 4,5-dihydropyrrolo[1,2-a]quinoxalines, methods for their preparation in a catalytic asymmetric fashion are limited.Therefore, it is highly desirable to develop efficient catalytic asymmetric methods for the synthesis of optically active 4,5-dihydropyrrolo[1,2-a]quinoxalines.
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