α-蒎烯和β-蒎烯是松节油的主要成分,因具有多种潜在的生物活性而受到广泛的关注。关于α-蒎烯和β-蒎烯及其衍生化合物药物活性的研究已有大量新的报道,但是全面系统的介绍仍然比较缺乏。因此,综述了近年来α-蒎烯和β-蒎烯药物活性的研究,以及利用α-蒎烯和β-蒎烯合成具有药物活性衍生化合物的研究进展,展望了α-蒎烯和β-蒎烯药物活性衍生化合物未来的研究发展方向。 α-pinene and β-pinene are the main components of turpentine, which have attracted extensive attention because of their potential biological activity. There have been a lot of new reports on the pharmacological activities of α-pinene and β-pinene and their derivatives, but a comprehensive and systematic introduction is still lacking. Therefore, in recent years, the research on the activity of α-pinene and β-pinene and the progress of synthesis of α-pinene and β-pinene derivatives with pharmacologically active compounds were reviewed. The effects of α-pinene and β- The Future Development of Pinene Derivatives.