TETRAHYDROQUINOLINE相关论文
以4-羟基香豆素和邻胺基苯甲醛为原料,高效合成了具有药物活性的3-位邻羟基苯甲酰基单取代的四氢喹啉衍生物.在乙醇溶剂中,反应经......
Kinetic Resolution of 2-Substituted 1,2-Dihydroquinolines by Rhodium-Catalyzed Asymmetric Hydroaryla
A highly efficient kinetic resolution of racemic 2-substituted 1,2-dihydroquinolines via Rh-catalyzed asymmetric hydroar......
本文发展了一种由当归内酯和邻氨基苯甲醛衍生物出发,经Aldol/Michael串联合环反应构建四氢呋喃并[3,2-b]喹啉-2(3H)-酮类化合物的......
Ball-milling Synthesis of Tetrahydroquinolines via‘One-pot’Three-component Diels-Alder Reaction Cata
We reported an economic and practical ball-milling method for the synthesis of tetrahydroquinoline derivatives via aone-......
Zirconyl Chloride Promoted Highly Efficient Domino Synthesis of New 1, 2, 3, 4-Tetrahydroquinoline D
The tetrahydroquinoline moiety is a structural feature of many natural products. By using a domino reaction of aromatic ......
Three-component one-pot synthesis of 1,2,3,4-tetrahydroquinoline derivatives in hexafluoroisopropano
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Zirconyl Chloride Promoted Highly Efficient Domino Synthesis of New 1, 2, 3, 4-Tetrahydroquinoline D
The tetrahydroquinoline moiety is a structural feature of many natural products. By using a domino reaction of aromatic ......
Three-component one-pot synthesis of 1,2,3,4-tetrahydroquinoline derivatives in hexafluoroisopropano
The one-pot aza-Diels-Alder reaction of substituted aromatic amines, ethyl glyoxylate and benzyl vinylcarbamate or N-ben......
四氢喹啉类化合物具有抑制血管舒张,抗肿瘤等活性^[1],也是更具特色的染料中间体^[2]。常用的合成方法有:取代的苯胺、醛和富电子烯烃......
目的寻找具有镇痛活性的新型四氢喹啉类化合物,探讨4-(1H-吡咯-2-基)-1,2,3,4-四氢喹啉类化合物镇痛作用的构效关系。方法以4-(1H-吡......
研究了在碘催化下亚胺与烯醇醚的反应,以较高的产率获得了预期的四氢喹啉产物。详细考察了催化剂的用量、亚胺的结构以及烯醇醚的......
本文合成了2—氨基—6—(β—羟乙基砜硫酸酯)苯骈噻唑和N—(β—羟乙基砜基乙基)-2,2,4,7—四甲基—1,2,3,4—四氢喹啉2个杂环中......