【摘 要】
:
The stereoselective synthesis of spiro-tetrahydroquinolines has been realized via cacade hydrogenative dearomatization[1] of quinoline and aza-Friedel-Crafts reaction.This methodology features ready a
【机 构】
:
State Key Laboratory of Organometallic Chemistry,Shanghai Institute of Organic Chemistry,Chinese Aca
【出 处】
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The 24th International Society of Heterocyclic Chemistry Con
论文部分内容阅读
The stereoselective synthesis of spiro-tetrahydroquinolines has been realized via cacade hydrogenative dearomatization[1] of quinoline and aza-Friedel-Crafts reaction.This methodology features ready available starting materials, operational simplicity and excellent yields.Further development of highly enantioselective reaction is currently underway in our laboratory.
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